Home Neuronal Signaling -GPCR & G Protein 5-HT Receptor 5-HT5 Antagonists

5-HT5 Antagonists

  • 5-HT1
  • 5-HT2
  • 5-HT3
  • 5-HT4
  • 5-HT6
  • 5-HT7
  • 5-HT5
N° Cat. Nom du produit Information Sélectif / Pan IC50 / Ki
S1283 Asenapine Asenapine is a high-affinity antagonist of serotonin, norepinephrine, dopamine and histamine receptors, used for the treatment of schizophrenia and acute mania associated with bipolar disorder. Pan 5-HT5A, pKi: 8.84
S1615 Risperidone Risperidone is a mutil-targeted antagonist for dopamine, serotonin, adrenergic and histamine receptors, used to treat schizophrenia and bipolar disorder. Pan 5-HT5A, Ki: 206 nM; 5-HT5A, Ki: 206 nM